Showing 3649–3664 of 5741 results

Guanabenz Acetate

Guanabenz Acetate is an selective agonist of α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor with pEC50 of 8.25, 7.01 and ~5, respectively.

Escitalopram Oxalate

Escitalopram Oxalate is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.

cholecalciferol (Vitamin D3)

Vitamin D3 is a form of vitamin D, binds and activates a H305F/H397Y mutant vitamin D receptor (VDR) with EC50 of 300 nM.

Levobupivacaine HCl

Levobupivacaine HCl, the pure S(-)-enantiomer of bupivacaine, is a reversible neuronal sodium channel inhibitor, used as a long-acting local anesthetic.

Erythromycin Ethylsuccinate

Erythromycin Ethylsuccinate, an oral macrolide antibiotic produced by Streptomyces erythreus, reversibly binds to the 50S ribosome of bacteria, and inhibits protein synthesis.

Ropivacaine HCl

Ropivacaine HCl is an anaesthetic agent and blocks impulse conduction in nerve fibres through inhibiting sodium ion influx reversibly.

Methyclothiazide

Methyclothiazide is a substituted benzothiadiazide, used to treat high blood pressure and fluid retention caused by various conditions including heart disease.

Retapamulin

Retapamulin is a topical antibiotic, which binds to both E. coli and S. aureus ribosomes with similar potencies with Kd of 3 nM.

Spironolactone

Spironolactone is a potent antagonist of the androgen receptor with IC50 of 77 nM.

Netilmicin Sulfate

Netilmicin Sulfate is a member of the aminoglycoside family of antibiotics.

Nabumetone

Nabumetone is a non-steroidal anti-inflammatory drug and its active metabolite inhibits the COX.

Valganciclovir HCl

Valganciclovir HCl is a prodrug for ganciclovir with antiviral activity used to treat cytomegalovirus infections.

Valdecoxib

Valdecoxib is a potent and selective inhibitor of COX-2 with IC50 of 5 nM.