Sodium Monofluorophosphate
Sodium Monofluorophosphate is a competitive inhibitor of pyruvate kinase and alkaline phosphatase with Ki of 3.4 mM and 69 μM, respectively, which also irreversibly inhibits phosphorylase phosphatase with Ki of 0.5 mM.
Showing 3697–3712 of 5738 results
Desloratadine
Desloratadine is a potent antagonist for human histamine H1 receptor with IC50 of 51 nM.
Ampiroxicam
Ampiroxicam is a nonselective cyclooxygenase inhibitor uesd as anti-inflammatory drug.
Acebutolol HCl
Acebutolol is a β-adrenergic receptors antagonist used in the treatment of hypertension, angina pectoris and cardiac arrhythmias.
Mirabegron
Mirabegron is a selective β3-adrenoceptor agonist with EC50 of 22.4 nM.
Pemirolast Potassium
Pemirolast potassium (BMY 26517) is a histamine H1 antagonist and mast cell stabilizer that acts as an antiallergic agent.
Pentamidine Isethionate
Pentamidine is an inhibitor of PRL Phosphatases and also inhibits synthesis of DNA, RNA and protein.
Clinafloxacin
Clinafloxacin is a fluoroquinolone that inhibits both DNA gyrase and topoisomerase IV dually in Streptococcus pneumoniae.
Ethambutol 2HCl
Ethambutol is a bacteriostatic antimycobacterial agent, which obstructs the formation of cell wall by inhibiting arabinosyl transferases.
Lithocholic Acid
Lithocholic acid is a toxic secondary bile acid, causes intrahepatic cholestasis, has tumor-promoting activity, its toxic effect can be protected after it activates the vitamin D receptor, PXR and FXR.
Sitagliptin Phosphate Monohydrate
Sitagliptin phosphate monohydrate is a potent inhibitor of DPP-IV with IC50 of 19 nM in Caco-2 cell extracts.
Cabozantinib Malate (XL184)
Cabozantinib malate (XL184) is the malate of Cabozantinib, a potent VEGFR2 inhibitor with IC50 of 0.035 nM and also inhibits c-Met, Ret, Kit, Flt-1/3/4, Tie2, and AXL with IC50 of 1.3 nM, 4 nM, 4.6 nM, 12 nM/11.3 nM/6 nM, 14.3 nM and 7 nM in cell-free assays, respectively.
Pergolide Mesylate
Pergolide Mesylate is an antiparkinsonian agent which functions as a dopaminergic agonist.
α-Santonin
α-santonin, a naturally occurring sesquiterpene lactone, is a potent antiparasitic agent.
(+)-α-Lipoic Acid
R(+)-α-lipoic acid, a physiological form of thioctic acid, is a strong antioxidant that relieves diabetic neuropathic symptoms. It shows superior antioxidative effects to its racemate.
Oxaceprol
Oxaceprol is an anti-inflammatory drug used in the treatment of osteoarthritis.