KG-501 (2-naphthol-AS-E-phosphate)

95.00 481.00 

KG-501 is a cAMP response element-binding protein (CREB) inhibitor that disrupts CREB-dependent transcription (Ki = 10 μM) and CREB:CBP interaction (Ki = 50 μM). It also disrupts phospho (Ser-133) CREB binding to KIX with a Ki of ≈90 μM, using concentrations of CREB that were within the linear range of the binding assay.

Clear

Additional information

Brand

Selleck Chemicals

CAS No.

18228-17-6

Molecular Weight

377.72

Signaling Pathway

Epigenetics

Target

Epigenetic Reader Domain

Storage

Store at -20°C