{"product_id":"sacubitril-valsartan-lcz696-s7678","title":"Sacubitril\/valsartan (LCZ696)","description":"\u003cp\u003e\u003cstrong\u003eSacubitril\/valsartan (LCZ696)\u003c\/strong\u003e is an inhibitor of Angiotensin Receptors used in studies of GPCR Signaling. It is especially relevant in cardiovascular models, where defined compound exposure can be linked to receptor-driven second-messenger signaling and desensitization dynamics.\u003c\/p\u003e\n\n\u003cp\u003eBy inhibiting Angiotensin Receptors, Sacubitril\/valsartan (LCZ696) can be used to examine receptor-driven second-messenger signaling and desensitization dynamics. The gpcr annotation adds relevance to GPCR pharmacology, ligand-binding, and signaling assays, together with downstream-response mapping in the same experimental setting. In cardiovascular models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.\u003c\/p\u003e\n\n\u003ch2\u003eResearch Applications\u003c\/h2\u003e\u003cul\u003e\n\u003cli\u003eTarget-focused assays involving Angiotensin Receptors\u003c\/li\u003e\n\u003cli\u003ePathway perturbation studies connected to GPCR Signaling\u003c\/li\u003e\n\u003cli\u003eConcentration-response inhibition and target-dependence studies\u003c\/li\u003e\n\u003cli\u003eGPCR pharmacology, ligand-binding, and signaling assays\u003c\/li\u003e\n\u003c\/ul\u003e\n\n\u003cp\u003eOverall, Sacubitril\/valsartan (LCZ696) is appropriate when a defined chemical perturbant is needed to connect Angiotensin Receptors with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cardiovascular models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.\u003c\/p\u003e","brand":"Selleck Chemicals","offers":[{"title":"5 mg","offer_id":57809530618201,"sku":"S7678-5MG","price":173.0,"currency_code":"EUR","in_stock":true},{"title":"25 mg","offer_id":57809530650969,"sku":"S7678-25MG","price":468.0,"currency_code":"EUR","in_stock":true},{"title":"1 g","offer_id":57809530683737,"sku":"S7678-1G","price":1641.0,"currency_code":"EUR","in_stock":true},{"title":"1 ml (10mM\/DMSO)","offer_id":57809530716505,"sku":"S7678-1ML\/DMSO","price":265.0,"currency_code":"EUR","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0923\/1011\/0553\/files\/lcz696-chemical-structure-s7678.gif?v=1776201704","url":"https:\/\/absource.de\/products\/sacubitril-valsartan-lcz696-s7678","provider":"Absource Diagnostics","version":"1.0","type":"link"}