Apararenone

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Selleck Chemicals

E1239-5MG

€175,00 EUR
€175,00 EUR
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Apararenone is an antagonist of Mineralocorticoid Receptor used in studies of Hormone Signaling. In practice, this places the compound in experiments that measure ligand-dependent transcriptional programs and endocrine regulation in cardiovascular and endocrinology models.

By blocking Mineralocorticoid Receptor, Apararenone can be used to examine ligand-dependent transcriptional programs and endocrine regulation. The nuclear receptor annotation adds relevance to reporter-gene, receptor-binding, and transcriptional assays, together with downstream-response mapping in the same experimental setting. In cardiovascular and endocrinology models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.

Research Applications

  • Target-focused assays involving Mineralocorticoid Receptor
  • Pathway perturbation studies connected to Hormone Signaling
  • Receptor-blockade and ligand-competition studies
  • Reporter-gene, receptor-binding, and transcriptional assays

Overall, Apararenone is appropriate when a defined chemical perturbant is needed to connect Mineralocorticoid Receptor with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cardiovascular and endocrinology models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.

Targets:
Mineralocorticoid Receptor
Target Class:
Nuclear Receptor
Pathways:
Hormone Signaling
Research Area:
Cardiovascular • Endocrinology
CAS No.:
945966-46-1
Molecular Weight:
364.39
Formula:
C₁₇H₁₇FN₂O₄S
Storage Temperature:
-20°C

For Research Use Only. Not intended for diagnostic or therapeutic use.
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The purchase of this product does not grant any license for commercial use, manufacturing, or clinical applications. The user is responsible for ensuring compliance with applicable laws and third-party rights.