AZD9496

1 1

Selleck Chemicals

S8372-2MG

€95,00 EUR
€95,00 EUR
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AZD9496 is an inhibitor of Estrogen/Progesterone Receptors and Estrogen Receptor used in studies of Hormone Signaling. In practice, this places the compound in experiments that measure ligand-dependent transcriptional programs and endocrine regulation in cancer and endocrinology models.

By inhibiting Estrogen/Progesterone Receptors and Estrogen Receptor, AZD9496 can be used to examine ligand-dependent transcriptional programs and endocrine regulation. The nuclear receptor annotation adds relevance to reporter-gene, receptor-binding, and transcriptional assays, together with downstream-response mapping in the same experimental setting. In cancer and endocrinology models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.

Research Applications

  • Target-focused assays involving Estrogen/Progesterone Receptors and Estrogen Receptor
  • Pathway perturbation studies connected to Hormone Signaling
  • Concentration-response inhibition and target-dependence studies
  • Reporter-gene, receptor-binding, and transcriptional assays

Overall, AZD9496 is appropriate when a defined chemical perturbant is needed to connect Estrogen/Progesterone Receptors and Estrogen Receptor with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cancer and endocrinology models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.

Targets:
Estrogen/Progesterone Receptors • Estrogen Receptor
Target Class:
Nuclear Receptor
Pathways:
Hormone Signaling
Research Area:
Cancer • Endocrinology
CAS No.:
1639042-08-2
Molecular Weight:
442.47
Formula:
C₂₅H₂₅F₃N₂O₂
SMILES:
CC1CC2=C(C(N1CC(C)(C)F)C3=C(C=C(C=C3F)C=CC(=O)O)F)NC4=CC=CC=C24
InChIKey:
DFBDRVGWBHBJNR-UHFFFAOYSA-N
PubChem:
86287635
Storage Temperature:
-20°C

For Research Use Only. Not intended for diagnostic or therapeutic use.
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