DC260126

1 1

Selleck Chemicals

S0742-5MG

€390,00 EUR
€390,00 EUR
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DC260126 is an antagonist of GPR and ERK1 used in studies of MAPK / ERK Signaling and GPCR Signaling. In practice, this places the compound in experiments that measure mitogenic kinase cascades, proliferation control, and differentiation-linked signaling and receptor-driven second-messenger signaling and desensitization dynamics in cancer and cell signaling models.

By blocking GPR and ERK1, DC260126 can be used to examine mitogenic kinase cascades, proliferation control, and differentiation-linked signaling and receptor-driven second-messenger signaling and desensitization dynamics. The gpcr annotation adds relevance to GPCR pharmacology, ligand-binding, and signaling assays, together with downstream-response mapping in the same experimental setting. In cancer and cell signaling models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.

Research Applications

  • Target-focused assays involving GPR and ERK1
  • Pathway perturbation studies connected to MAPK / ERK Signaling and GPCR Signaling
  • Receptor-blockade and ligand-competition studies
  • GPCR pharmacology, ligand-binding, and signaling assays

Overall, DC260126 is appropriate when a defined chemical perturbant is needed to connect GPR and ERK1 with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cancer and cell signaling models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.

Targets:
GPR • ERK1
Target Class:
GPCR
Pathways:
MAPK / ERK Signaling • GPCR Signaling
Research Area:
Cancer • Cell Signaling
CAS No.:
346692-04-4
Molecular Weight:
307.38
Formula:
C₁₆H₁₈FNO₂S
SMILES:
CCCCC1=CC=C(C=C1)NS(=O)(=O)C2=CC=C(C=C2)F
Storage Temperature:
-20°C

For Research Use Only. Not intended for diagnostic or therapeutic use.
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The purchase of this product does not grant any license for commercial use, manufacturing, or clinical applications. The user is responsible for ensuring compliance with applicable laws and third-party rights.