Eprosartan
Selleck Chemicals
SKU:E4951-5MG
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Eprosartan is an antagonist of Angiotensin Receptors and Sphingosine Kinases used in studies of GPCR Signaling and Metabolic Signaling. It is especially relevant in cardiovascular, immunology, and inflammation models, where defined compound exposure can be linked to receptor-driven second-messenger signaling and desensitization dynamics and metabolic regulation, energy sensing, and enzyme-linked homeostasis.
By blocking Angiotensin Receptors and Sphingosine Kinases, Eprosartan can be used to examine receptor-driven second-messenger signaling and desensitization dynamics and metabolic regulation, energy sensing, and enzyme-linked homeostasis. The gpcr annotation adds relevance to GPCR pharmacology, ligand-binding, and signaling assays, together with downstream-response mapping in the same experimental setting. In cardiovascular, immunology, and inflammation models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.
Research Applications
- Target-focused assays involving Angiotensin Receptors and Sphingosine Kinases
- Pathway perturbation studies connected to GPCR Signaling and Metabolic Signaling
- Receptor-blockade and ligand-competition studies
- GPCR pharmacology, ligand-binding, and signaling assays
Overall, Eprosartan is appropriate when a defined chemical perturbant is needed to connect Angiotensin Receptors and Sphingosine Kinases with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cardiovascular, immunology, and inflammation models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.
- Targets:
- Angiotensin Receptors • Sphingosine Kinases
- Target Class:
- GPCR
- Pathways:
- GPCR Signaling • Metabolic Signaling
- Research Area:
- Cardiovascular • Immunology • Inflammation • Metabolism
- CAS No.:
- 133040-01-4
- Molecular Weight:
- 424.51
- Formula:
- C₂₃H₂₄N₂O₄S
- SMILES:
- CCCCc1ncc(/C=C(\Cc2cccs2)C(=O)O)n1Cc1ccc(C(=O)O)cc1
- InChIKey:
- OROAFUQRIXKEMV-LDADJPATSA-N
- PubChem:
- 5281037
- Storage Temperature:
- -20°C
For Research Use Only. Not intended for diagnostic or therapeutic use.
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