MI-136

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Selleck Chemicals

S7815-5MG

€193,00 EUR
€193,00 EUR
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MI-136 is an inhibitor of Histone Methyltransferases and Transferases used in studies of Epigenetic Regulation and Hormone Signaling and related signaling programs. In practice, this places the compound in experiments that measure chromatin-state control, histone modification, and transcriptional regulation and ligand-dependent transcriptional programs and endocrine regulation in cancer, endocrinology, and epigenetics models.

By inhibiting Histone Methyltransferases and Transferases, MI-136 can be used to examine chromatin-state control, histone modification, and transcriptional regulation and ligand-dependent transcriptional programs and endocrine regulation. The epigenetic regulator annotation adds relevance to chromatin, epigenetic, and gene-expression profiling, together with downstream-response mapping in the same experimental setting. In cancer, endocrinology, and epigenetics models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.

Research Applications

  • Target-focused assays involving Histone Methyltransferases and Transferases
  • Pathway perturbation studies connected to Epigenetic Regulation and Hormone Signaling and related signaling programs
  • Concentration-response inhibition and target-dependence studies
  • Chromatin, epigenetic, and gene-expression profiling

Overall, MI-136 is appropriate when a defined chemical perturbant is needed to connect Histone Methyltransferases and Transferases with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cancer, endocrinology, and epigenetics models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.

Targets:
Histone Methyltransferases • Transferases
Target Class:
Epigenetic Regulator
Pathways:
Epigenetic Regulation • Hormone Signaling • Metabolic Signaling
Research Area:
Cancer • Endocrinology • Epigenetics • Metabolism
CAS No.:
1628316-74-4
Molecular Weight:
470.51
Formula:
C₂₃H₂₁F₃N₆S
SMILES:
C1CN(CCC1NC2=C3C=C(SC3=NC=N2)CC(F)(F)F)CC4=CC5=C(C=C4)NC(=C5)C#N
Storage Temperature:
-20°C

For Research Use Only. Not intended for diagnostic or therapeutic use.
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