Pelabresib (CPI-0610)

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Selleck Chemicals

S7853-5MG

€293,00 EUR
€293,00 EUR
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Pelabresib (CPI-0610) is an inhibitor of BET and MYC used in studies of Cell Cycle Regulation and Epigenetic Regulation. In practice, this places the compound in experiments that measure checkpoint control, mitotic progression, and proliferation timing and chromatin-state control, histone modification, and transcriptional regulation in cancer and epigenetics models.

By inhibiting BET and MYC, Pelabresib (CPI-0610) can be used to examine checkpoint control, mitotic progression, and proliferation timing and chromatin-state control, histone modification, and transcriptional regulation. The epigenetic regulator annotation adds relevance to chromatin, epigenetic, and gene-expression profiling, together with downstream-response mapping in the same experimental setting. In cancer and epigenetics models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.

Research Applications

  • Target-focused assays involving BET and MYC
  • Pathway perturbation studies connected to Cell Cycle Regulation and Epigenetic Regulation
  • Concentration-response inhibition and target-dependence studies
  • Chromatin, epigenetic, and gene-expression profiling

Overall, Pelabresib (CPI-0610) is appropriate when a defined chemical perturbant is needed to connect BET and MYC with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cancer and epigenetics models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.

Targets:
BET • MYC
Target Class:
Epigenetic Regulator
Pathways:
Cell Cycle Regulation • Epigenetic Regulation
Research Area:
Cancer • Epigenetics
CAS No.:
1380087-89-7
Molecular Weight:
365.81
Formula:
C₂₀H₁₆ClN₃O₂
SMILES:
CC1=NOC2=C1C3=CC=CC=C3C(=NC2CC(=O)N)C4=CC=C(C=C4)Cl
Storage Temperature:
-20°C

For Research Use Only. Not intended for diagnostic or therapeutic use.
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