Picfeltarraenin IA
Selleck Chemicals
SKU:S9138-1MG
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Picfeltarraenin IA is an inhibitor of AChR and EGFR and related targets used in studies of PI3K-Akt-mTOR Signaling and MAPK / ERK Signaling and related signaling programs. It is especially relevant when investigators need a named chemical input and interpretable readouts connected to growth-factor signaling, survival control, and nutrient-sensing outputs and mitogenic kinase cascades, proliferation control, and differentiation-linked signaling in cancer, cell signaling, and metabolism models.
By inhibiting AChR and EGFR and related targets, Picfeltarraenin IA can be used to examine growth-factor signaling, survival control, and nutrient-sensing outputs and mitogenic kinase cascades, proliferation control, and differentiation-linked signaling. The kinase annotation adds relevance to biochemical kinase assays, phospho-signaling studies, and selectivity profiling, together with downstream-response mapping in the same experimental setting. In cancer, cell signaling, and metabolism models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.
Research Applications
- Target-focused assays involving AChR and EGFR and related targets
- Pathway perturbation studies connected to PI3K-Akt-mTOR Signaling and MAPK / ERK Signaling and related signaling programs
- Concentration-response inhibition and target-dependence studies
- Biochemical kinase assays, phospho-signaling studies, and selectivity profiling
Overall, Picfeltarraenin IA is appropriate when a defined chemical perturbant is needed to connect AChR and EGFR and related targets with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cancer, cell signaling, and metabolism models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.
- Targets:
- AChR • EGFR • PI3K
- Target Class:
- Kinase
- Pathways:
- PI3K-Akt-mTOR Signaling • MAPK / ERK Signaling • Neurotransmission
- Research Area:
- Cancer • Cell Signaling • Metabolism • Neuroscience
- CAS No.:
- 97230-47-2
- Molecular Weight:
- 762.92
- Formula:
- C₄₁H₆₂O₁₃
- SMILES:
- CC1C(C(C(C(O1)OC2C(C(COC2OC3CCC4C(=CCC5C4(C(=O)CC6(C5(CC(C6C7(C(=O)C=C(O7)C(C)C)C)O)C)C)C)C3(C)C)O)O)O)O)O
- Storage Temperature:
- -20°C
For Research Use Only. Not intended for diagnostic or therapeutic use.
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