Tefinostat (CHR-2845)

1 1

Selleck Chemicals

E1554-1MG

€193,00 EUR
€193,00 EUR
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Tefinostat (CHR-2845) is an inhibitor of HDAC used in studies of Epigenetic Regulation. In practice, this places the compound in experiments that measure chromatin-state control, histone modification, and transcriptional regulation in cancer and epigenetics models.

By inhibiting HDAC, Tefinostat (CHR-2845) can be used to examine chromatin-state control, histone modification, and transcriptional regulation. The epigenetic regulator annotation adds relevance to chromatin, epigenetic, and gene-expression profiling, together with downstream-response mapping in the same experimental setting. In cancer and epigenetics models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.

Research Applications

  • Target-focused assays involving HDAC
  • Pathway perturbation studies connected to Epigenetic Regulation
  • Concentration-response inhibition and target-dependence studies
  • Chromatin, epigenetic, and gene-expression profiling

Overall, Tefinostat (CHR-2845) is appropriate when a defined chemical perturbant is needed to connect HDAC with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cancer and epigenetics models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.

Targets:
HDAC
Target Class:
Epigenetic Regulator
Pathways:
Epigenetic Regulation
Research Area:
Cancer • Epigenetics
CAS No.:
914382-60-8
Molecular Weight:
495.61
Formula:
C₂₈H₃₇N₃O₅
PubChem:
15940949
Storage Temperature:
-20°C

For Research Use Only. Not intended for diagnostic or therapeutic use.
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The purchase of this product does not grant any license for commercial use, manufacturing, or clinical applications. The user is responsible for ensuring compliance with applicable laws and third-party rights.