Tinostamustine (EDO-S101)

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Selleck Chemicals

S8769-1MG

€144,00 EUR
€144,00 EUR
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Tinostamustine (EDO-S101) is an inhibitor of HDAC used in studies of Epigenetic Regulation. It is especially relevant in cancer and epigenetics models, where defined compound exposure can be linked to chromatin-state control, histone modification, and transcriptional regulation.

By inhibiting HDAC, Tinostamustine (EDO-S101) can be used to examine chromatin-state control, histone modification, and transcriptional regulation. The epigenetic regulator annotation adds relevance to chromatin, epigenetic, and gene-expression profiling, together with downstream-response mapping in the same experimental setting. In cancer and epigenetics models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.

Research Applications

  • Target-focused assays involving HDAC
  • Pathway perturbation studies connected to Epigenetic Regulation
  • Concentration-response inhibition and target-dependence studies
  • Chromatin, epigenetic, and gene-expression profiling

Overall, Tinostamustine (EDO-S101) is appropriate when a defined chemical perturbant is needed to connect HDAC with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cancer and epigenetics models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.

Targets:
HDAC
Target Class:
Epigenetic Regulator
Pathways:
Epigenetic Regulation
Research Area:
Cancer • Epigenetics
CAS No.:
1236199-60-2
Molecular Weight:
415.36
Formula:
C₁₉H₂₈Cl₂N₄O₂
SMILES:
CN1C2=C(C=C(C=C2)N(CCCl)CCCl)N=C1CCCCCCC(=O)NO
InChIKey:
GISXTRIGVCKQBX-UHFFFAOYSA-N
PubChem:
46836227
Storage Temperature:
-20°C

For Research Use Only. Not intended for diagnostic or therapeutic use.
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