XMD8-92

1 1

Selleck Chemicals

S7525-10MG

€144,00 EUR
€144,00 EUR
Sold out
Shipping calculated at checkout.
Supplier
Size
View full details

XMD8-92 is an inhibitor of ERK and BET used in studies of MAPK / ERK Signaling and Epigenetic Regulation. In practice, this places the compound in experiments that measure mitogenic kinase cascades, proliferation control, and differentiation-linked signaling and chromatin-state control, histone modification, and transcriptional regulation in cancer, cell signaling, and epigenetics models.

By inhibiting ERK and BET, XMD8-92 can be used to examine mitogenic kinase cascades, proliferation control, and differentiation-linked signaling and chromatin-state control, histone modification, and transcriptional regulation. The kinase annotation adds relevance to biochemical kinase assays, phospho-signaling studies, and selectivity profiling, together with downstream-response mapping in the same experimental setting. In cancer, cell signaling, and epigenetics models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.

Research Applications

  • Target-focused assays involving ERK and BET
  • Pathway perturbation studies connected to MAPK / ERK Signaling and Epigenetic Regulation
  • Concentration-response inhibition and target-dependence studies
  • Biochemical kinase assays, phospho-signaling studies, and selectivity profiling

Overall, XMD8-92 is appropriate when a defined chemical perturbant is needed to connect ERK and BET with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cancer, cell signaling, and epigenetics models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.

Targets:
ERK • BET
Target Class:
Kinase
Pathways:
MAPK / ERK Signaling • Epigenetic Regulation
Research Area:
Cancer • Cell Signaling • Epigenetics
CAS No.:
1234480-50-2
Molecular Weight:
474.55
Formula:
C₂₆H₃₀N₆O₃
SMILES:
CCOC1=C(C=CC(=C1)N2CCC(CC2)O)NC3=NC=C4C(=N3)N(C5=CC=CC=C5C(=O)N4C)C
Storage Temperature:
-20°C

For Research Use Only. Not intended for diagnostic or therapeutic use.
Products may be subject to intellectual property rights.

The purchase of this product does not grant any license for commercial use, manufacturing, or clinical applications. The user is responsible for ensuring compliance with applicable laws and third-party rights.